教育背景
1998/09-2002/06,西南民族大学,应用化学,学士
2002/09-2005/06,四川大学,有机化学,硕士
2007/09-2011/06,西南大学,药用资源化学,博士
工作经历
2005/07-至今, 西南大学,药学院,教师
项目课题经历
承担的主要科研项目
1.国家自然科学基金青年项目,21602180,以NF-κB为靶点的大环蒽醌类似物的合成与抗炎活性构效关系研究,2017/01-2019/12,20万,主持
2.西南大学基本科研业务费专项资金项目,XDJK2016C071,大环蒽醌类IκB激酶抑制剂的合成和抗炎活性研究,2016/01-2017/12,5万元,主持
3. 西南大学博士基金,SWU111064,大黄酰胺类衍生物的合成与降糖活性研究,2012/01-2015/12,5万元,主持
4. 西南大学基本科研业务费专项资金项目,XDJK2011C050,具有抗炎活性的大黄酸衍生物的设计、合成和活性研究,2011/09-2014/09,5万元,主持
5. 西南大学科研基金项目,SWU208040,大黄素类衍生物的合成与生物活性研究,2009/01-2010/12,2万,主持
6. 国家自然科学基金面上项目,21477098,多氯联苯醌引起的氧化应激相关信号转导与神经毒性作用机制及抗氧化剂干预,2015/01-2018/12,88万,参加
7. 国家科技重大专项课题,2010ZX09401-306-3-10,黄连治疗糖尿病型高血脂并发症中药新药研究,2010/01-2012/12,57万,参加
论文、成果、著作等
代表论文
(1)Xiaokang Zhu, Mingdong Jiang, Erqun Song, Xiaoji Jiang, Yang Song*. Selenium dediciency sensitizes the skin for UVB-induced oxidative damage and inflammation which involved the activation of p38 MAPK signaling. Food Chem. Toxicol., 2015, 75, 139-145
(2) Xiaokang Zhu, Xiaoli Ye, Liu Song, Yonghuang Luo, Qing Tang, Yanan Jin, Xuegang Li*. Synthesis and hypoglycemic activity evaluation of rhein amide derivatives. Med. Chem. Res., 2013, 22, 2228-2234.
(3) Xiaokang Zhu, Xiaoli Ye, Lujiang Yuan, Yangping Ding, Baoshun Zhang, Xuegang Li*. Synthesis and hypoglycemic activity evaluation of 7-alkyoxyl- rhein. Med. Chem. Res., 2012, 21(4), 421-427.
(4) 朱小康,叶小利,袁吕江,朱家颖,丁阳平,李学刚*. 微波辐射下6-烷氧基大黄酸的合成及抑菌活性研究.有机化学, 2010, 30(9), 1335-1341
(5) 朱小康,杨玉金,田晋红,李学刚*. N-( 卤代芳酰)-亚肼基二噻烷的合成及抑菌活性. 西南大学学报,2010, 32(5):74-77
(6) Yuxin Wanga, Linyao Li, Yawen Wang, Xiaokang Zhu, Mingdong Jiang, Erqun Song, Yang Song. New application of the commercial sweetener rebaudioside a as a hepatoprotective candidate: Induction of the Nrf2 signaling pathway. Eur. J. Pharmacol., 2018, 822: 128-137
(7) David A. Leigh*, Vanesa Marcos, Tugrul Nalbantoglu, Iñigo J. Vitorica -Yrezabal, F. Tuba Yasar, Xiaokang Zhu. Pyridyl-Acyl Hydrazone Rotaxanes and Molecular Shuttles. J. Am. Chem. Soc., 2017, 139, 7104- 7109.
(8) Yangping Ding, Xiaoli Ye, Jiaying Zhu, Xiaokang Zhu, Xuegang Li*, Bingcan Chen*. Structural modification of berberine alkaloid and their hypoglycemic activity. J. Funct. Foods, 2014, 7: 229-237
(9) Tao Wang, XiaoKang Zhu, XuTing Xue, DaYang Wu*. Hydrogel sheets of chitosan, honey and gelatin as burn wound dressings. Carbohydr Polym,2012, 88(1), 75-83
(10) Xingguo Tian, Erqun Song, Ruxian Pi, Xiaokang Zhu, Lichao Liu, Xiaoyan Ma, Hui Dong, Jing Liu, Yang Song*. Polychlorinated biphenyls and their different level metabolites as inhibitors of glutathione S-transferase isoenzymes. Chem-Biol Interact., 2012, 198(s1-3):1-8
(11) Xiaoli Ye, Kai He, Xiaokang Zhu, Baoshun Zhang, Xin Chen, Jun Yi, Xuegang Li*. Synthesis and antihyperlipidemic efficiency of berberine-based HMG-CoA reductase inhibitor. Med. Chem. Res., 2012, 21: 1353- 1362
专利、著作版权等
李学刚,朱小康,叶小利,3-烷氧基-6-羧基大黄酸或其可药用盐及其制备方法和应用,2013.1.31,中国,ZL200910104466.5.
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