教育背景
2009年9月至2014年6月攻读中国药科大学药物化学博士学位。2014年7月毕业并获理学博士学位,
工作经历
项目课题经历
1. 国家自然科学基金面上项目,31870325,基于微管蛋白抑制的抗乳腺癌多药耐药天然呋喃[2,3-b]喹啉类化合物的发现与结构修饰研究,2019/01-2022/12,在研,主持。
2. 国家自然科学基金青年基金项目,31500277,基于拓扑异构酶II抑制的白鲜皮中抗肺癌喹诺酮的结构修饰与构效关系研究,2016/01-2018/12,在研,主持。
3. 中央高校基本业务经费重点项目,ZY20180117041,基于天然呋喃喹啉类化合物设计合成兼具抗菌及抗肿瘤活性的新型Topo II抑制剂,2018/7-2020/6,在研,主持。
4. 横向课题,校合2018-中12,保健食品生物利用度、产品功能及毒理学研究,2018/06-2021/05,在研,主持。
5. 横向课题,校合2017-中56,陕西安康普欣药业联合建设中药配方颗粒标准化工程中心,2018/03-2020/02,在研,主持。
6. 横向课题,山东罗欣药业盐酸美金刚原料结构测试试验(校合2018-中4)、盐酸头孢他美酯原料结构确证(校合2017-中14)及原料结构测试试验(校合2017-中52,校合2019-中015),2017/01-2019/12,在研,主持。
7. 广西艾滋病防治研究重点实验室开放课题基金,gklapt201701,基于HIV整合酶抑制的天然抗艾滋病病毒4-喹啉酮类药物的筛选与结构修饰研究,2018/01-2020/12,在研,主持。
8. 区域性高发肿瘤早期防治研究重点实验室开放课题基金,GK2015-TKF02,白鲜皮中抗肝癌呋喃喹诺酮的发现与构效关系研究,2016/1-2017/12,结题,主持。
9. 陕西省肿瘤精准医学重点实验室开放课题,KLTPM-SX2022-B3,兼具抗菌和肿瘤活性的天然呋喃喹啉类DNA拓扑异构酶II抑制剂的筛选与结构修饰研究,2018/1-2020/12,在研,主持。
10. 科技部“重大新药创制”重大科技专项课题、2011ZX09307-002、中药化学与活性成分库的子课题中药化学成分库建设、参加。
论文、成果、著作等
1.Sun Jianbo,Qu Wei, Wang Pei, Wu Feihua*, Wang Liying, Liang Jingyu*. Degraded limonoids and quinoline alkaloids from Dictamnus angustifoliusG. Don ex Sweet. and their anti-platelet aggregation activity. Fitoterapia, 2013, 90:209-213.
2.Sun Jianbo#*,Jiang Neng#, Lv Mengying, Tang Benqin, Wang Pei, Liang Jingyu, Chen Li*.Anstifolines A and B, two dimeric furoquinoline alkaloids from the root bark of Dictamnus angustifolius. RSC Advances, 2016, 47(28):22550-22554.
3.Sun Jianbo, Wang Xinzhi, Wang Pei, Li Linzhen, Qu Wei*, Liang Jingyu*. Antimicrobial, antioxidant and cytotoxic properties of essential oil from Dictamnus angustifolius. Journal of Ethnopharmacology, 2015, 159:296-300.
4.Wang Bing, Li Qiangqiang, Shi Wei, Chen Li*, Sun Jianbo*. Design, synthesis, and cytotoxic evaluation of novel furo[2,3-b]quinoline derivatives. Chemical Biology & Drug Design. 2018, 91(4):957-961.
5.Sun Jianbo#, Jiang Neng#, Lv Mengying, Wang Pei, Xu Fengguo, Liang Jingyu*, Qu Wei*. Limonoids from the root bark of Dictamnus angustifolius: potent neuroprotective agent with biometal chelation, halting copper redox cycling properties. RSC Advances, 2015, 5:24750-24757.
6.Sun Jianbo#, Tang Benqin#, Li Qiangqiang, Wang Bing, Liang Jingyu*, Chen Li*.Cytotoxic limonoids from the root bark of Dictamnus angustifolius. Fitoterapia, 2016, 115:92-95.
7.Lv Mengying, Tian Yuan, Zhang Zunjian, Xu Fengguo*, Sun Jianbo*. Plant metabolomics driven chemical and biological comparison of the root bark of Dictamnus dasycarpus and Dictamnus angustifolius. 2015, RSC Advances, 5(20):15700-15708.
8.Lv Mengying, Xu Ping, Tian Yuan, Liang Jingyu, Gao Yiqiao, Xu Fengguo, Zhang Zunjian*, Sun Jianbo*. Medicinal uses, phytochemistry and pharmacology of the genus Dictamnus (Rutaceae). Journal of Ethnopharmacology, 2015, 171: 247-263.
9.Li Qixing, Zou Pian, Sun Jianbo*, Chen Li*. O2-(2,4-dinitrophenyl) diazeniumdiolates derivatives: Design, synthesis, cytotoxic evaluation and reversing MDR in HepG-2/ADR cells. European Journal of Medicinal Chemistry, 2018, 143:732-744.
10.Bao Na#, Ou Jinfeng#, Xu Manyi, Guan Fuqin, Shi Wei, Sun Jianbo*, Chen Li*. Novel NO-releasing plumbagin derivatives: Design, synthesis and evaluation of antiproliferative activity. European Journal of Medicinal Chemistry, 2017, 137:88-95.
11.Bao Na#, Ou Jinfeng#, Li Na, Zou Pian, Sun Jianbo*, Chen Li*. Novel anticancer hybrids from diazen-1-ium-1,2-diolate nitric oxide donor and ROS inducer plumbagin: Design, synthesis and biological evaluations. European Journal of Medicinal Chemistry, 2018, 154:1-8.
12.Shi Wei, Hu Jinglin, Bao Na, Li Dongang, Chen Li*, Sun Jianbo*. Design, synthesis and cytotoxic activities of scopoletin-isoxazole and scopoletin-pyrazole hybrids. Bioorganic and Medicinal Chemistry Letters, 2017, 27(2):147-151.
13.Shi Wei, Zhang Jinlu, Bao Na, Guan Fuqin, Chen Li*, Sun Jianbo*.Design, synthesis and cytotoxic evaluation of novel scopoletin derivatives. Chemical Biology & Drug Design. 2018, 91(2):641-646.
14.Liu Yan, Wang Tingting, Ling Yong, Bao Na, Shi Wei, Chen Li*, Sun Jianbo*. Design, synthesis and cytotoxic evaluation of nitric oxide-releasing derivatives of isosteviol. Chemical Biology & Drug Design. 2017, 90(3):473-477.
15.Liu Jinhong, Zhu Zifei, Tang Jia, Lin Qinghua, Chen Li*, Sun Jianbo*. Design and Synthesis of NO-releasing Betulinic Acid Derivatives as Potential Anticancer Agents. Anti-cancer Agents in Medicinal Chemistry, 2017, 17:241-249.
16.Wang Pei#, Sun Jianbo#, Gao Enze, Zhao Yunli, Qu Wei, Yu Zhiguo*. Simultaneous determination of limonin, dictamnine, obacunone and fraxinellone in rat plasma by a validated UHPLC-MS/MS and its application to a pharmacokinetic study after oral administration of Cortex Dictamni extract. Journal of Chromatography B, 2013, 928(0):44-51.
17.Wang Pei#, Sun Jianbo#, Xu Jingyao, Gao Enze, Yan Qin, Qu Wei, Zhao Yunli, Yu Zhiguo*. Pharmacokinetics, tissue distribution and excretion study of dictamnine, a major bioactive component from the root bark of Dictamnus dasycarpus Turcz. (Rutaceae). Journal of Chromatography B, 2013, 942-943:1-8.
专利、著作版权等
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